PPARgamma Antagonist III, G3335 – CAS 36099-95-3 – Calbiochem

REF : 516566-50MG
Marca : Sigma-Aldrich
Descrição :PPARgamma Antagonist III, G3335 - CAS 36099-95-3 - Calbiochem The PPARgamma Antagonist III, G3335, also referenced under CAS 36099-95-3, controls the biological activity of PPARgamma.
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Descrição detalhada : A cell-permeable dipeptide that acts as a selective and reversible PPARgamma antagonist (KD ~8 µM). Shown to inhibit the agonist activity of Rosiglitazone (100 nM) in a dose-dependent manner (IC50 = 31.9 µM) in transfected COS-7 cells., A cell-permeable dipeptide that acts as a selective and reversible PPARgamma antagonist (KD = ~ 8 µM). Shown to inhibit the agonist activity of Rosiglitazone (100 nM) in a dose-dependent manner (IC50 = 31.9 µM) in transfected COS-7 cells.
Sinónimos : PPARgamma Antagonist III, G3335 - CAS 36099-95-3 - Calbiochem; H-Trp-Glu-OH
Fórmula molecula r: C16H19N3O5
Armazenamento : 2-8C; 2-8C; 2-8C
Embalagem : 1X50MG