TAPI-0 – CAS 143457-40-3 – Calbiochem

REF : 579050-1MG
Marca : Sigma-Aldrich
Descrição :TAPI-0 - CAS 143457-40-3 - Calbiochem TAPI-0, CAS 143457-40-3, is a hydroxamate-based inhibitor of collagenase, gelatinase, and TACE (TNF-alpha converting enzyme/ADAM17; IC?? = 100 nM).
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Descrição detalhada : A hydroxymate-based inhibitor of collagenase, gelatinase, and TACE [(TNF-alpha convertase; ADAM17 (IC50 = 100 nM)]. Blocks spontaneous and PMA-induced release of TNF-alpha from transfected COS-7 cells., A hydroxamate-based inhibitor of collagenase, gelatinase, and TACE (TNF-alpha converting enzyme/ADAM17; IC50 = 100 nM). Blocks spontaneous and PMA-induced release of TNF-alpha in transfected COS 7 cells.
Sinónimos : TAPI-0 - CAS 143457-40-3 - Calbiochem; N-(R)-[2-(Hydroxyaminocarbonyl)methyl]-4-methylpentanoyl-L-naphthylalanyl-L-alanine Amide, TNF-alpha Protease Inhibitor-0
Fórmula molecula r: C24H32N4O5
Armazenamento : -20C
Embalagem : 1X1MG