DAPK Inhibitor – CAS 315694-89-4 – Calbiochem

REF : 324788-10MG
Marca : Sigma-Aldrich
Descrição :DAPK Inhibitor - CAS 315694-89-4 - Calbiochem The DAPK Inhibitor, also referenced under CAS 315694-89-4, controls the biological activity of DAPK.
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Descrição detalhada : An oxazalone compound that acts as a potent, ATP-competitive, and highly selective death-associated protein kinase (DAPK) inhibitor (IC50 = 69 and 225 nM against DAPK1 and DAPK3, respectively, with 10 µM ATP), while exhibiting much reduced or no activity against a panel of 48 other kinases even at concentrations as high as 10 µM.
Sinónimos : DAPK Inhibitor - CAS 315694-89-4 - Calbiochem; (4 Z)-4-(3-Pyridylmethylene)-2-styryl-oxazol-5-one, Death-Associated Protein Kinase Inhibitor; (4Z)-4-(3-Pyridylmethylene)-2-styryl-oxazol-5-one, Death-Associated Protein Kinase Inhibitor
Fórmula molecula r: C17H12N2O2
Armazenamento : 2-8C; 2-8C; 2-8C
Embalagem : 1X10MG