FGF/PDGF/VEGF RTK Inhibitor – CAS 144335-37-5 – Calbiochem
REF : 341610-5MG
Marca : Sigma-Aldrich
Descrição :FGF/PDGF/VEGF RTK Inhibitor - CAS 144335-37-5 - Calbiochem The FGF/PDGF/VEGF RTK Inhibitor, also referenced under CAS 144335-37-5, controls the biological activity of FGF/PDGF/VEGF RTK. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
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Categoria : Small Molecules
Descrição detalhada : A cell-permeable benzimidazolo-hydroquinolinone compound that acts as a potent, reversible, ATP-competitive inhibitor against PDGFRβ, FGFR-1, and VEGFR-2 (IC50 = 20, 90, and 240 nM, respectively) and effectively suppresses VEGF-stimulated proliferation of HMVECs (EC50 = 420 nM).
Sinónimos : FGF/PDGF/VEGF RTK Inhibitor - CAS 144335-37-5 - Calbiochem; 4-Hydroxy-3-benzimidazol-2-ylhydroquinolin-2-one, PDGFR Tyrosine Kinase Inhibitor XVII, VEGFR Tyrosine Kinase Inhibitor XXX, VEGFR2 Kinase Inhibitor XXVIII; PDGFR Tyrosine Kinase Inhibitor XVII, 4-Hydroxy-3-benzimidazol-2-ylhydroquinolin-2-one, VEGFR Tyrosine Kinase Inhibitor XXX, VEGFR2 Kinase Inhibitor XXVIII
Fórmula molecula r: C16H11N3O2
Armazenamento : 2-8C; 2-8C; 2-8C
Embalagem : 1X5MG
Sinónimos : FGF/PDGF/VEGF RTK Inhibitor - CAS 144335-37-5 - Calbiochem; 4-Hydroxy-3-benzimidazol-2-ylhydroquinolin-2-one, PDGFR Tyrosine Kinase Inhibitor XVII, VEGFR Tyrosine Kinase Inhibitor XXX, VEGFR2 Kinase Inhibitor XXVIII; PDGFR Tyrosine Kinase Inhibitor XVII, 4-Hydroxy-3-benzimidazol-2-ylhydroquinolin-2-one, VEGFR Tyrosine Kinase Inhibitor XXX, VEGFR2 Kinase Inhibitor XXVIII
Fórmula molecula r: C16H11N3O2
Armazenamento : 2-8C; 2-8C; 2-8C
Embalagem : 1X5MG
