InSolution NF-kappaB Activation Inhibitor – Calbiochem

REF : 481407-1MG
Marca : Sigma-Aldrich
Descrição :InSolution NF-kappaB Activation Inhibitor - Calbiochem The InSolution NF-kappaB Activation Inhibitor controls the biological activity of NF-kappaB. This small molecule/inhibitor is primarily used for Inflammation/Immunology applications.
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Descrição detalhada : A cell-permeable quinazoline compound that acts as a potent inhibitor of NF-kappaB transcriptional activation (IC50 = 11 nM in Jurkat cells) and LPS-induced TNF-alpha production (IC50 = 7 nM in murine splenocytes). Does not exhibit cellular cytotoxicity even at concentrations as high as 10 µM. Reported to exhibit anti-inflammatory effects on carregeenin-induced paw edema in rats.
Sinónimos : InSolution NF-kappaB Activation Inhibitor - Calbiochem
Fórmula molecula r: C22H20N4O
Armazenamento : 2-8C; 2-8C; 2-8C; 2-8C
Embalagem : 1X1MG