Ketanserin Tartrate – CAS 83846-83-7 – Calbiochem
REF : 5062710001
Marca : Sigma-Aldrich
Descrição :
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Categoria : Small Molecules
Descrição detalhada : A selective 5-HT2A serotonin receptor antagonist with weak adrenergic receptor blocking properties. Strong affinity for 5-HT2AR (Ki = 1.49 nM) relative to other family members like 5-HT2BR (Ki = 740 nM) and 5-HT2CR (Ki = 59 nM). Often used in conjunction with SB 206553 to distinguish 5-HT2AR and 5-HT2CR activity., A selective 5-HT2A serotonin receptor antagonist with weak adrenergic receptor blocking properties. Strong affinity for 5-HT2AR (Ki = 1.49 nM) relative to other family members like 5-HT2BR (Ki = 740 nM) and 5-HT2CR (Ki = 59 nM). Often used in conjunction with SB 206553 to distinguish 5-HT2AR and 5-HT2CR activity.
Sinónimos : Ketanserin Tartrate - CAS 83846-83-7 - Calbiochem; 5-HT 2A Serotonin Receptor Antagonist, Ketanserin, R 41 468
Fórmula molecula r: C22H22FN3O3 · xC4H6O6
Armazenamento : 2-8C; 2-8C; 2-8C
Embalagem : 1X1EA
Sinónimos : Ketanserin Tartrate - CAS 83846-83-7 - Calbiochem; 5-HT 2A Serotonin Receptor Antagonist, Ketanserin, R 41 468
Fórmula molecula r: C22H22FN3O3 · xC4H6O6
Armazenamento : 2-8C; 2-8C; 2-8C
Embalagem : 1X1EA
