L-745,870 Trihydrochloride – CAS 158985-00-3 – Calbiochem

REF : 5058800001
Marca : Sigma-Aldrich
Categoria :
Descrição detalhada : Selective D4 receptor antagonist with excellent brain penetration. Displays an affinity (Ki) of 0.4 nM for human D4 receptors with >1000-fold binding selectivity over D2 and D3 receptors. Does not block agonist-induced activation of GIRK currents. It is used frequently in retinal and CNS studies of D4 modulation.
Sinónimos : L-745,870 Trihydrochloride - CAS 158985-00-3 - Calbiochem; Dopamine D? receptor Antagonist, L-745,870 trihydrochloride, L-745870, L745870
Fórmula molecula r: C18H19ClN4 · 3HCl
Armazenamento : 2-8C; 2-8C; 2-8C
Embalagem : 1X1EA