Stearoyl-CoA Desaturase 1 Inhibitor, MF-438 – Calbiochem
REF : 569406-10MG
Marca : Sigma-Aldrich
Descrição :Stearoyl-CoA Desaturase 1 Inhibitor, MF-438 - Calbiochem Stearoyl-CoA Desaturase 1 Inhibitor, MF-438, CAS 921605-87-0, is a cell-permeable inhibitor of Stearoyl-CoA Desaturase 1 (SCD1; IC50 of 2.3 nM).
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Categoria : Small Molecules
Descrição detalhada : A cell-permeable, thiadiazole-pyridazine compound that acts as an inhibitor of Stearoyl-CoA Desaturase 1 (SCD1) with an IC50 of 2.3 nM. In vivo, it exhibits an ED50 of 1-3 mg/kg, p.o., in mouse liver PD assays.
Sinónimos : Stearoyl-CoA Desaturase 1 Inhibitor, MF-438 - Calbiochem; 2-methyl-5-(6-(4-(2-(trifluoromethyl)phenoxy)piperidin-1-yl)pyridazin-3-yl)-1,3,4-thiadiazole
Fórmula molecula r: C19H18F3N5OS
Armazenamento : 2-8C; 2-8C
Embalagem : 1X10MG
Sinónimos : Stearoyl-CoA Desaturase 1 Inhibitor, MF-438 - Calbiochem; 2-methyl-5-(6-(4-(2-(trifluoromethyl)phenoxy)piperidin-1-yl)pyridazin-3-yl)-1,3,4-thiadiazole
Fórmula molecula r: C19H18F3N5OS
Armazenamento : 2-8C; 2-8C
Embalagem : 1X10MG
