Cytisine

Descrição detalhada : Cytisine was found to be more effective than nicotine-replacement therapy in helping smokers to quit smoking. It is an ?4 ?2 nicotinic receptor partial agonist. It is a plant alkaloid which is commercially extracted for use as a smoking cessation medication. Preparation of nicotine partial agonist cytisine via "in situ" Stille or Suzuki biaryl pyridine coupling has been reported. Cytisine is a competitive partial agonist at ?4 subunit-containing nicotinic acetylcholine (nACh) receptors while at homomeric ?7-nACh receptors it behaves as a full agonist with a relatively lower potency., Cystine ((1R,5S)-1,2,3,4,5,6-hexahydro-1,5-methano-8H-pyrido[1,2a][1,5]diazocin-8-one) displays classical antidepressant action in various animal models of antidepressant efficacy. Infrared and Raman spectral studies suggest that it has two stable conformers.
Sinónimos : (-)-Cytisine; (1R,5S)-1,2,3,4,5,6-Hexahydro-1,5-methano-8H-pyrido[1,2a][1,5]diazocin-8-one; (1S,9S)-3,11-Diazatricyclo[7.3.1.03,8]trideca-5,7-dien-4-one; Baptitoxin; Laburnin; Sophorine; Ulexine
Fórmula molecula r: C11H14N2O
Armazenamento : Room Temperature
Embalagem : 1X100MG