SR95531 (Gabazine) – CAS 104104-50-9 – Calbiochem

Descrição detalhada : A selective, competitive antagonist of GABAA receptor (IC50 = 440 nM) that does not affect pentobarbitone or etomidate- induced currents even at high concentrations (~100 µM). Also shown to block glycine receptors, but with low affinity (Kb = 190 µM)., A selective, competitive antagonist of GABAA receptor (IC50 = 440 nM) that does not affect pentobarbitone or etomidate- induced currents even at high concentrations (~100 mM). Also shown to block glycine receptors, but with low affinity (Kb = 190 mM).
Sinónimos : SR95531 (Gabazine) - CAS 104104-50-9 - Calbiochem; GABA A Receptor Antagonist, SR-95531, Gabazine, SR95531, SR 95531; GABAA Receptor Antagonist, SR-95531, Gabazine, SR95531, SR 95531
Fórmula molecula r: C15H17N3O3 · xHBr
Armazenamento : 2-8C; 2-8C
Embalagem : 1X1EA